Skip to contents

Savić, Marina [Editor]; Mernyák, Erzsébet [Editor]; Ajdukovic, Jovana [Editor]; Jovanović-Šanta, Suzana [Editor]

Steroid Compounds with Potential Biological Activity

View online
Schließen

Access

https://directory.doabooks.org/handle/20.500.12854/132467

Show more show less

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Basel: MDPI - Multidisciplinary Digital Publishing Institute, 2023
Burinsky, D.; Williams, J.; Thornquest, A. Jr.; Sides, S.

Mass Spectral Fragmentation Reactions of 4‐Azasteroids

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Wiley, 2004

Published in: ChemInform
Liang, T.; Cheung, A.; Reynolds, G.F.; Rasmusson, G.H.

323 4-Azasteroids as inhibitors of 5α-reductase

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Elsevier BV, 1983

Published in: Journal of Steroid Biochemistry
Ruda, Marcus C.; Bergman, Jan; Koehler, Konrad; Liu, Ye

A SOLUTION-PHASE PROCEDURE FOR THE PREPARATION OF 4-AZASTEROID MIMETICS

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Walter de Gruyter GmbH, 2003

Published in: Heterocyclic Communications
Burinsky, David J.; Williams, Jon D.; Thornquest, Alan D.; Sides, Scott L.

Mass spectral fragmentation reactions of a therapeutic 4-azasteroid and related compounds

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

American Chemical Society (ACS), 2001

Published in: Journal of the American Society for Mass Spectrometry
Di Salle, E.; Briatico, G.; Giudici, D.; Ornati, G.; Nesi, M.; Panzeri, A.

17β-acylurea derivatives of 4-azasteroids as inhibitors of testosterone 5α-reductase

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Elsevier BV, 1992

Published in: The Journal of Steroid Biochemistry and Molecular Biology
Brooks, Jerry R.; Primka, Raymond L.; Bel-man, Charles; Krupa, David A.; Reynolds, Glenn F.; Rasmusson, Gary H.

Topical anti-androgenicity of a new 4-azasteroid in the hamster

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Elsevier BV, 1991

Published in: Steroids
Vermeulen, A.; Giagulli, V. A.; De Schepper, P.; Buntinx, A.; Stoner, E.

Hormonal effects of an orally active 4‐azasteroid inhibitor of 5α‐reductase in humans

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Wiley, 1989

Published in: The Prostate
Brooks, J.R.; Berman, C.; Primka, R.L.; Reynolds, G.F.; Rasmusson, G.H.

5α-Reductase inhibitory and anti-androgenic activities of some 4-azasteroids in the rat

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Elsevier BV, 1986

Published in: Steroids
Mitchell, Helen J.; Dankulich, William P.; Hartman, George D.; Prueksaritanont, Thomayant; Schmidt, Azriel; Vogel, Robert L.; Bai, Chang; McElwee-Witmer, Sheila; Zhang, Hai Z.; Chen, Fang; Leu, Chih-Tai; Kimmel, Donald B.; Ray, William J.; Nantermet, Pascale; Gentile, Michael A.; Duggan, Mark E.; Meissner, Robert S.

Design, Synthesis, and Biological Evaluation of 16-Substituted 4-Azasteroids as Tissue-Selective Androgen Receptor Modulators (SARMs)

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

American Chemical Society (ACS), 2009

Published in: Journal of Medicinal Chemistry
Taylor, Matthew F.; Bhattacharyya, Anjan K.; Rajagopalan, Krishnan; Hiipakka, Richard; Liao, Shutsung; Collins, Delwood C.

Photoaffinity labeling of rat steroid 5α-reductase (isozyme-1) by a benzophenone derivative of a 4-methyl-4-azasteroid

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Elsevier BV, 1996

Published in: Steroids
Kim, Sujeong; Kim, Yong-ung; Ma, Eunsook

Synthesis and 5α-Reductase Inhibitory Activity of C21 Steroids Having 1,4-diene or 4,6-diene 20-ones and 4-Azasteroid 20-Oximes

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

MDPI AG, 2011

Published in: Molecules
Tian, Gaochao; Haffner, Curt D.

Linear Relationships between the Ligand Binding Energy and the Activation Energy of Time-dependent Inhibition of Steroid 5α-Reductase by Δ1-4-Azasteroids

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Elsevier BV, 2001

Published in: Journal of Biological Chemistry
Grisenti, Paride; Magni, Ambrogio; Olgiati, Vincenzo; Manzocchi, Ada; Ferraboschi, Patrizia; Villani, Vincenzo; Pucciariello, Rachele; Celotti, Fabio

Substrate interaction with 5α-reductase enzyme: influence of the 17β-chain chirality in the mechanism of action of 4-azasteroid inhibitors

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Elsevier BV, 2001

Published in: Steroids
Tolman, Richard L.; Aster, Susan; Bakshi, Raman K.; Bergman, Jeffrey P.; Bull, Herb G.; Chang, Benedict; Cimis, George; Dolenga, Michael P.; Durette, Phillippe; Ellsworth, Kenneth; Esser, Craig; Graham, Donald W.; Hagmann, William K.; Harris, Georgianna; Kopka, Ihor; Lanza, Thomas; Patel, Gool; Polo, Scott; Rasmusson, Gary H.; Sahoo, Soumya; Toney, Jeffrey H.; Von Langen, Derek; Witzel, Bruce

4-AZASTEROIDS AS 5α-REDUCTASE INHIBITORS: IDENTIFICATION OF 4,7β-DIMETHYL-4-AZA-5α-CHOLESTAN-3-ONE (MK-386) AS A SCALP ISOZYME SELECTIVE INHIBITOR

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Elsevier BV, 1995

Published in: European Journal of Medicinal Chemistry
Bakshi, Raman K.; Patel, Gool F.; Rasmusson, Gary H.; Baginsky, Walter F.; Cimis, George; Ellsworth, Kenneth; Chang, Benedict; Bull, Herb; Tolman, Richard L.; Harris, Georgianna S.

4,7.beta.-Dimethyl-4-azacholestan-3-one (MK-386) and Related 4-Azasteroids as Selective Inhibitors of Human Type 1 5.alpha.-Reductase

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

American Chemical Society (ACS), 1994

Published in: Journal of Medicinal Chemistry
Back, Thomas G.; Chau, Joseph H.-L.; Dyck, Brian P.; Gladstone, Patricia L.

The synthesis of some novel N-chloro-Δ1-4-azasteroids by efficient N-chlorination of azasteroid lactams with trichloroisocyanuric acid

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Canadian Science Publishing, 1991

Published in: Canadian Journal of Chemistry
GUARNA, A.; OCCHIATO, E. G.; MACHETTI, F.; MARRUCCI, A.; DANZA, G.; SERIO, M.; PAOLI, P.

ChemInform Abstract: 19‐Nor‐10‐azasteroids, a New Class of Steroid 5α‐Reductase Inhibitors. Part 2. X‐Ray Structure, Molecular Modeling, Conformational Analysis of 19‐Nor‐10‐azasteroids and Comparison with 4‐Azasteroids and 6‐Azasteroids

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Wiley, 1998

Published in: ChemInform
Guarna, Antonio; Occhiato, Ernesto G.; Machetti, Fabrizio; Marrucci, Alessandro; Danza, Giovanna; Serio, Mario; Paoli, Paola

19-Nor-10-azasteroids, a New Class of Steroid 5α-Reductase Inhibitors. 2. X-ray Structure, Molecular Modeling, Conformational Analysis of 19-Nor-10-azasteroids and Comparison with 4-Azasteroids and 6-Azasteroids

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

American Chemical Society (ACS), 1997

Published in: Journal of Medicinal Chemistry
Constanzer, M.L; Chavez, C.M; Matuszewski, B.K; Carlin, J; Graham, D

Low level determination of a novel 4-azasteroid and its carboxylic acid metabolite in human plasma and semen using high-performance liquid chromatography with atmospheric pressure chemical ionization tandem mass spectrometry

View online
Schließen

Access

Close

Bookmarks

You can manage bookmarks using lists, please log in to your user account for this.

Elsevier BV, 1997

Published in: Journal of Chromatography B: Biomedical Sciences and Applications

You did not find what you were looking for?

Purchase suggestion
Are you missing something you need for your research? If you have any suggestions please share them here.

Interlibrary Loan
Please search and order your favorite title in the Interlibrary Loan Portal.

Search in field:

Recently searched for:

You did not find what you were looking for?

> Year of publication

Year of publication