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  1. Marciniak, Monika [Author]; Mróz, Piotr [Author]; Napolitano, Valeria [Author]; Kalel, Vishal C. [Author]; Fino, Roberto [Author]; Pykacz, Emilia [Author]; Schliebs, Wolfgang [Author]; Plettenburg, Oliver [Author]; Erdmann, Ralf [Author]; Sattler, Michael [Author]; Popowicz, Grzegorz M. [Author]; Dawidowski, Maciej [Author]

    Development of novel PEX5-PEX14 protein-protein interaction (PPI) inhibitors based on an oxopiperazine template - [published Version]

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    Amsterdam [u.a.] : Elsevier Science, 2023

    Published in: European Journal of Medicinal Chemistry 258 (2023) ; European Journal of Medicinal Chemistry

  3. Fino, Roberto [Author]; Lenhart, Dominik [Author]; Kalel, Vishal C. [Author]; Softley, Charlotte A. [Author]; Napolitano, Valeria [Author]; Byrne, Ryan [Author]; Schliebs, Wolfgang [Author]; Dawidowski, Maciej [Author]; Erdmann, Ralf [Author]; Sattler, Michael [Author]; Schneider, Gisbert [Author]; Plettenburg, Oliver [Author]; Popowicz, Grzegorz M. [Author]

    Computer-Aided Design and Synthesis of a New Class of PEX14 Inhibitors: Substituted 2,3,4,5-Tetrahydrobenzo[F][1,4]oxazepines as Potential New Trypanocidal Agents

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    Hannover: Gottfried Wilhelm Leibniz Universität Hannover, 2021 ; Hannover: Technische Informationsbibliothek (TIB), 2021

    Published in: Journal of Chemical Information and Modeling ; 61 (2021), Nr. 10, S. 5256-5268

  4. Fino, Roberto [Author]; Lenhart, Dominik [Author]; Kalel, Vishal C. [Author]; Softley, Charlotte A. [Author]; Napolitano, Valeria [Author]; Byrne, Ryan [Author]; Schliebs, Wolfgang [Author]; Dawidowski, Maciej [Author]; Erdmann, Ralf [Author]; Sattler, Michael [Author]; Schneider, Gisbert [Author]; Plettenburg, Oliver [Author]; Popowicz, Grzegorz M. [Author]

    Computer-Aided Design and Synthesis of a New Class of PEX14 Inhibitors: Substituted 2,3,4,5-Tetrahydrobenzo[F][1,4]oxazepines as Potential New Trypanocidal Agents - [published Version]

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    Washington, DC : American Chemical Society, 2021

    Published in: Journal of Chemical Information and Modeling 61 (2021), Nr. 10 ; Journal of Chemical Information and Modeling

  5. Dawidowski, Maciej [Author]; Kalel, Vishal C. [Author]; Napolitano, Valeria [Author]; Fino, Roberto [Author]; Schorpp, Kenji [Author]; Emmanouilidis, Leonidas [Author]; Lenhart, Dominik [Author]; Ostertag, Michael [Author]; Kaiser, Marcel [Author]; Kolonko, Marta [Author]; Tippler, Bettina [Author]; Schliebs, Wolfgang [Author]; Dubin, Grzegorz [Author]; Mäser, Pascal [Author]; Tetko, Igor V. [Author]; Hadian, Kamyar [Author]; Plettenburg, Oliver [Author]; Erdmann, Ralf [Author]; Sattler, Michael [Author]; Popowicz, Grzegorz M. [Author]

    Structure-Activity Relationship in Pyrazolo[4,3- c]pyridines, First Inhibitors of PEX14-PEX5 Protein-Protein Interaction with Trypanocidal Activity

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    Hannover: Gottfried Wilhelm Leibniz Universität Hannover, 2019 ; Hannover: Technische Informationsbibliothek (TIB), 2019

    Published in: Journal of Medicinal Chemistry (formerly: Journal of Medicinal and Pharmaceutical Chemistry) ; 63 (2020), Nr. 2, S. 847-879

  6. Dawidowski, Maciej [Author]; Kalel, Vishal C. [Author]; Napolitano, Valeria [Author]; Fino, Roberto [Author]; Schorpp, Kenji [Author]; Emmanouilidis, Leonidas [Author]; Lenhart, Dominik [Author]; Ostertag, Michael [Author]; Kaiser, Marcel [Author]; Kolonko, Marta [Author]; Tippler, Bettina [Author]; Schliebs, Wolfgang [Author]; Dubin, Grzegorz [Author]; Mäser, Pascal [Author]; Tetko, Igor V. [Author]; Hadian, Kamyar [Author]; Plettenburg, Oliver [Author]; Erdmann, Ralf [Author]; Sattler, Michael [Author]; Popowicz, Grzegorz M. [Author]

    Structure-Activity Relationship in Pyrazolo[4,3- c]pyridines, First Inhibitors of PEX14-PEX5 Protein-Protein Interaction with Trypanocidal Activity - [published Version]

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    Washington, DC : ACS, 2019

    Published in: Journal of Medicinal Chemistry (formerly: Journal of Medicinal and Pharmaceutical Chemistry) 63 (2020), Nr. 2 ; Journal of Medicinal Chemistry (formerly: Journal of Medicinal and Pharmaceutical Chemistry)

  7. Bonatto, Vinicius; Batista, Pedro Henrique Jatai; Cianni, Lorenzo; De Vita, Daniela; Silva, Daniel G.; Cedron, Rodrigo; Tezuka, Daiane Y.; de Albuquerque, Sérgio; Moraes, Carolina Borsoi; Franco, Caio Haddad; Lameira, Jerônimo; Leitão, Andrei; Montanari, Carlos A.

    On the intrinsic reactivity of highly potent trypanocidal cruzain inhibitors

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    Royal Society of Chemistry (RSC), 2020

    Published in: RSC Medicinal Chemistry

  8. Bayliss, Tracy; Robinson, David A.; Smith, Victoria C.; Brand, Stephen; McElroy, Stuart P.; Torrie, Leah S.; Mpamhanga, Chido; Norval, Suzanne; Stojanovski, Laste; Brenk, Ruth; Frearson, Julie A.; Read, Kevin D.; Gilbert, Ian H.; Wyatt, Paul G.

    Design and Synthesis of Brain Penetrant Trypanocidal N-Myristoyltransferase Inhibitors

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    American Chemical Society (ACS), 2017

    Published in: Journal of Medicinal Chemistry

  14. Pauli, Ivani; Rezende Jr., Celso de O.; Slafer, Brian W.; Dessoy, Marco A.; de Souza, Mariana L.; Ferreira, Leonardo L. G.; Adjanohun, Abraham L. M.; Ferreira, Rafaela S.; Magalhães, Luma G.; Krogh, Renata; Michelan-Duarte, Simone; Del Pintor, Ricardo Vaz; da Silva, Fernando B. R.; Cruz, Fabio C.; Dias, Luiz C.; Andricopulo, Adriano D.

    Multiparameter Optimization of Trypanocidal Cruzain Inhibitors With In Vivo Activity and Favorable Pharmacokinetics

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    Frontiers Media SA, 2022

    Published in: Frontiers in Pharmacology

  19. Chacón-Vargas, Karla; Nogueda-Torres, Benjamin; Sánchez-Torres, Luvia; Suarez-Contreras, Erick; Villalobos-Rocha, Juan; Torres-Martinez, Yuridia; Lara-Ramirez, Edgar; Fiorani, Giulia; Krauth-Siegel, R.; Bolognesi, Maria; Monge, Antonio; Rivera, Gildardo

    Trypanocidal Activity of Quinoxaline 1,4 Di-N-oxide Derivatives as Trypanothione Reductase Inhibitors

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    MDPI AG, 2017

    Published in: Molecules

  20. Avelar, Leandro A. A.; Camilo, Cristian D.; de Albuquerque, Sérgio; Fernandes, William B.; Gonçalez, Cristiana; Kenny, Peter W.; Leitão, Andrei; McKerrow, James H.; Montanari, Carlos A.; Orozco, Erika V. Meñaca; Ribeiro, Jean F. R.; Rocha, Josmar R.; Rosini, Fabiana; Saidel, Marta E.

    Molecular Design, Synthesis and Trypanocidal Activity of Dipeptidyl Nitriles as Cruzain Inhibitors

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    Public Library of Science (PLoS), 2015

    Published in: PLOS Neglected Tropical Diseases