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  2. Lancelot, Julien [Author]; Caby, Stéphanie [Author]; Dubois-Abdesselem, Florence [Author]; Jung, Manfred [Author]

    Schistosoma mansoni sirtuins: characterization and potential as chemotherapeutic targets

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    San Francisco: Public Library of Science, 2013

    Published in: PLOS Neglected Tropical Diseases ; 7, 9 (2013), e2428

  3. Pagliazzo, Lucile [Author]; Caby, Stéphanie [Author]; Lancelot, Julien [Author]; Salomé-Desnoulez, Sophie [Author]; Saliou, Jean-Michel [Author]; Heimburg, Tino [Author]; Chassat, Thierry [Author]; Cailliau, Katia [Author]; Sippl, Wolfgang [Author]; Vicogne, Jérôme [Author]; Pierce, Raymond J. [Author]

    Histone deacetylase 8 interacts with the GTPase SmRho1 in Schistosoma mansoni

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    2021

    Published in: Public Library of Science: PLoS neglected tropical diseases ; 15(2021), 11, Artikel-ID e0009503

  4. Kalinin, Dmitrii V. [Author]; Jana, Sunit Kumar [Author]; Pfafenrot, Maxim [Author]; Chakrabarti, Alokta [Author]; Melesina, Jelena [Author]; Shaik, Tajith B. [Author]; Lancelot, Julien [Author]; Pierce, Raymond J. [Author]; Sippl, Wolfgang [Author]; Romier, Christophe [Author]; Jung, Manfred [Author]; Holl, Ralph [Author]

    Structure‐based design, synthesis, and biological evaluation of triazole‐based smHDAC8 inhibitors

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    2020

    Published in: ChemMedChem ; 15(2020), 7, Seite 571-584

  5. Kalinin, Dmitrii V. [Author]; Jana, Sunit Kumar [Author]; Pfafenrot, Maxim [Author]; Chakrabarti, Alokta [Author]; Melesina, Jelena [Author]; Shaik, Tajith B. [Author]; Lancelot, Julien [Author]; Pierce, Raymond J. [Author]; Sippl, Wolfgang [Author]; Romier, Christophe [Author]; Jung, Manfred [Author]; Holl, Ralph [Author]

    Structure‐based design, synthesis, and biological evaluation of triazole‐based smHDAC8 inhibitors

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    Weinheim: Wiley-VCH, 2020

    Published in: ChemMedChem ; 15, 7 (2020), 571-584

  6. Marek, Martin [Author]; Shaik, Tajith B. [Author]; Heimburg, Tino [Author]; Chakrabarti, Alokta [Author]; Lancelot, Julien [Author]; Ramos-Morales, Elizabeth [Author]; Da Veiga, Cyrielle [Author]; Kalinin, Dmitrii [Author]; Melesina, Jelena [Author]; Robaa, Dina [Author]; Schmidtkunz, Karin [Author]; Suzuki, Takayoshi [Author]; Holl, Ralph [Author]; Ennifar, Eric [Author]; Pierce, Raymond J. [Author]; Jung, Manfred [Author]; Sippl, Wolfgang [Author]; Romier, Christophe [Author]

    Characterization of histone deacetylase 8 (HDAC8) selective inhibition reveals specific active site structural and functional determinants

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    October 22, 2018

    Published in: Journal of medicinal chemistry ; 61(2018), 22, Seite 10000-10016

  7. Simoben, Conrad V. [Author]; Robaa, Dina [Author]; Chakrabarti, Alokta [Author]; Schmidtkunz, Karin [Author]; Marek, Martin [Author]; Lancelot, Julien [Author]; Kannan, Srinivasaraghavan [Author]; Melesina, Jelena [Author]; Shaik, Tajith B. [Author]; Pierce, Raymond J. [Author]; Romier, Christophe [Author]; Jung, Manfred [Author]; Sippl, Wolfgang [Author]

    A novel class of Schistosoma mansoni histone deacetylase 8 (HDAC8) inhibitors identified by structure-based virtual screening and in vitro testing

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    Basel: MDPI, 2018

    Published in: Molecules ; 23, 3 (2018), article no. 566

  8. Stolfa, Diana A. [Author]; Marek, Martin [Author]; Lancelot, Julien [Author]; Hauser, Alexander-Thomas [Author]; Walter, Alexandra [Author]; Leproult, Emeline [Author]; Melesina, Jelena [Author]; Rumpf, Tobias [Author]; Wurtz, Jean-Marie [Author]; Cavarelli, Jean [Author]; Sippl, Wolfgang [Author]; Pierce, Raymond J. [Author]; Romier, Christophe [Author]; Jung, Manfred [Author]

    Molecular basis for the antiparasitic activity of a mercaptoacetamide derivative that inhibits histone deacetylase 8 (HDAC8) from the human pathogen schistosoma mansoni

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    Amsterdam [u.a.]: Elsevier, 2014

    Published in: Journal of molecular biology ; Volume 426, Issue 20 (2014), pages 3442-3453

  9. Coutinho Carneiro, Vitor [Author]; Abreu da Silva, Isabel Caetano de [Author]; Amaral, Murilo Sena [Author]; Pereira, Adriana S. A. [Author]; Silveira, Gilbert Oliveira [Author]; Pires, David da Silva [Author]; Verjovski-Almeida, Sergio [Author]; Dekker, Frank J. [Author]; Rotili, Dante [Author]; Mai, Antonello [Author]; Lopes-Torres, Eduardo José [Author]; Robaa, Dina [Author]; Sippl, Wolfgang [Author]; Pierce, Raymond J. [Author]; Borrello, M. Teresa [Author]; Ganesan, A. [Author]; Lancelot, Julien [Author]; Thiengo, Silvana [Author]; Fernandez, Monica Ammon [Author]; Vicentino, Amanda Roberta Revoredo [Author]; Mourão, Marina Moraes [Author]; Coelho, Fernanda Sales [Author]; Fantappié, Marcelo Rosado [Author]

    Pharmacological inhibition of lysine-specific demethylase 1 (LSD1) induces global transcriptional deregulation and ultrastructural alterations that impair viability in Schistosoma mansoni

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    2020

    Published in: Public Library of Science: PLoS neglected tropical diseases ; 14 (2020,7), Artikel e0008332, 29 Seiten

  12. Valentin, Sarah; Arsevska, Elena; Mercier, Alize; Falala, Sylvain; Rabatel, Julien; Lancelot, Renaud; Roche, Mathieu

    Human Language Technology. Challenges for Computer Science and Linguistics: PADI-web: An Event-Based Surveillance System for Detecting, Classifying and Processing Online News

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    Springer International Publishing, 2020

    Published in: Human Language Technology. Challenges for Computer Science and Linguistics (2020), Seite 87-101

  15. Morel, Marion; Vanderstraete, Mathieu; Cailliau, Katia; Lescuyer, Arlette; Lancelot, Julien; Dissous, Colette

    Compound library screening identified Akt/PKB kinase pathway inhibitors as potential key molecules for the development of new chemotherapeutics against schistosomiasis

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    Elsevier BV, 2014

    Published in: International Journal for Parasitology: Drugs and Drug Resistance, 4 (2014) 3, Seite 256-266

  17. Vanderstraete, Mathieu; Gouignard, Nadège; Cailliau, Katia; Morel, Marion; Lancelot, Julien; Bodart, Jean-François; Dissous, Colette

    Dual Targeting of Insulin and Venus Kinase Receptors of Schistosoma mansoni for Novel Anti-schistosome Therapy

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    Public Library of Science (PLoS), 2013

    Published in: PLoS Neglected Tropical Diseases, 7 (2013) 5, Seite e2226

  20. Lancelot, Julien; Caby, Stéphanie; Dubois-Abdesselem, Florence; Vanderstraete, Mathieu; Trolet, Jacques; Oliveira, Guilherme; Bracher, Franz; Jung, Manfred; Pierce, Raymond J.

    Schistosoma mansoni Sirtuins: Characterization and Potential as Chemotherapeutic Targets

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    Public Library of Science (PLoS), 2013

    Published in: PLoS Neglected Tropical Diseases, 7 (2013) 9, Seite e2428