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  1. Theoclitou, Maria-Elena; Aquila, Brian; Block, Michael H.; Brassil, Patrick J.; Castriotta, Lillian; Code, Erin; Collins, Michael P.; Davies, Audrey M.; Deegan, Tracy; Ezhuthachan, Jayachandran; Filla, Sandra; Freed, Ellen; Hu, Haiqing; Huszar, Dennis; Jayaraman, Muthusamy; Lawson, Deborah; Lewis, Paula M; Nadella, Murali V. P.; Oza, Vibha; Padmanilayam, Maniyan; Pontz, Timothy; Ronco, Lucienne; Russell, Daniel; Whitston, David;

    Discovery of (+)-N-(3-Aminopropyl)-N-[1-(5-benzyl-3-methyl-4-oxo-[1,2]thiazolo[5,4-d]pyrimidin-6-yl)-2-methylpropyl]-4-methylbenzamide (AZD4877), a Kinesin Spindle Protein Inhibitor and Potential Anticancer Agent

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    American Chemical Society (ACS), 2011

    Published in: Journal of Medicinal Chemistry, 54 (2011) 19, Seite 6734-6750

  2. Casás‐Selves, Matias; Zhang, Andrew X.; Dowling, James E.; Hallén, Stefan; Kawatkar, Aarti; Pace, Nicholas J.; Denz, Christopher R.; Pontz, Timothy; Garahdaghi, Farzin; Cao, Qing; Sabirsh, Alan; Thakur, Kumar; O'Connell, Nichole; Hu, Jun; Cornella‐Taracido, Iván; Weerapana, Eranthie; Zinda, Michael; Goodnow, Robert A.; Castaldi, M. Paola

    Cover Picture: Target Deconvolution Efforts on Wnt Pathway Screen Reveal Dual Modulation of Oxidative Phosphorylation and SERCA2 (ChemMedChem 12/2017)

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    Wiley, 2017

    Published in: ChemMedChem, 12 (2017) 12, Seite 860-860

  3. Casás‐Selves, Matias; Zhang, Andrew X.; Dowling, James E.; Hallén, Stefan; Kawatkar, Aarti; Pace, Nicholas J.; Denz, Christopher R.; Pontz, Timothy; Garahdaghi, Farzin; Cao, Qing; Sabirsh, Alan; Thakur, Kumar; O'Connell, Nichole; Hu, Jun; Cornella‐Taracido, Iván; Weerapana, Eranthie; Zinda, Michael; Goodnow, Robert A.; Castaldi, M. Paola

    Target Deconvolution Efforts on Wnt Pathway Screen Reveal Dual Modulation of Oxidative Phosphorylation and SERCA2

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    Wiley, 2017

    Published in: ChemMedChem, 12 (2017) 12, Seite 917-924

  4. Vasbinder, Melissa M.; Aquila, Brian; Augustin, Martin; Chen, Huawei; Cheung, Tony; Cook, Donald; Drew, Lisa; Fauber, Benjamin P.; Glossop, Steve; Grondine, Michael; Hennessy, Edward; Johannes, Jeffrey; Lee, Stephen; Lyne, Paul; Mörtl, Mario; Omer, Charles; Palakurthi, Sangeetha; Pontz, Timothy; Read, Jon; Sha, Li; Shen, Minhui; Steinbacher, Stefan; Wang, Haixia; Wu, Allan;

    Discovery and Optimization of a Novel Series of Potent Mutant B-RafV600E Selective Kinase Inhibitors

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    American Chemical Society (ACS), 2013

    Published in: Journal of Medicinal Chemistry, 56 (2013) 5, Seite 1996-2015

  5. Dowling, James E.; Alimzhanov, Marat; Bao, Larry; Block, Michael H.; Chuaqui, Claudio; Cooke, Emma L.; Denz, Christopher R.; Hird, Alex; Huang, Shan; Larsen, Nicholas A.; Peng, Bo; Pontz, Timothy W.; Rivard-Costa, Caroline; Saeh, Jamal Carlos; Thakur, Kumar; Ye, Qing; Zhang, Tao; Lyne, Paul D.

    Structure and Property Based Design of Pyrazolo[1,5-a]pyrimidine Inhibitors of CK2 Kinase with Activity in Vivo

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    American Chemical Society (ACS), 2013

    Published in: ACS Medicinal Chemistry Letters, 4 (2013) 8, Seite 800-805

  6. Dowling, James E.; Chuaqui, Claudio; Pontz, Timothy W.; Lyne, Paul D.; Larsen, Nicholas A.; Block, Michael H.; Chen, Huawei; Su, Nancy; Wu, Allan; Russell, Daniel; Pollard, Hannah; Lee, John W.; Peng, Bo; Thakur, Kumar; Ye, Qing; Zhang, Tao; Brassil, Patrick; Racicot, Vicki; Bao, Larry; Denz, Christopher R.; Cooke, Emma

    Potent and Selective Inhibitors of CK2 Kinase Identified through Structure-Guided Hybridization

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    American Chemical Society (ACS), 2012

    Published in: ACS Medicinal Chemistry Letters, 3 (2012) 4, Seite 278-283