• Media type: E-Article
  • Title: Structure-Based Optimization of Potent, Selective, and Orally Bioavailable CDK8 Inhibitors Discovered by High-Throughput Screening
  • Contributor: Czodrowski, Paul; Mallinger, Aurélie; Wienke, Dirk; Esdar, Christina; Pöschke, Oliver; Busch, Michael; Rohdich, Felix; Eccles, Suzanne A.; Ortiz-Ruiz, Maria-Jesus; Schneider, Richard; Raynaud, Florence I.; Clarke, Paul A.; Musil, Djordje; Schwarz, Daniel; Dale, Trevor; Urbahns, Klaus; Blagg, Julian; Schiemann, Kai
  • Published: American Chemical Society (ACS), 2016
  • Published in: Journal of Medicinal Chemistry
  • Extent: 9337-9349
  • Language: English
  • DOI: 10.1021/acs.jmedchem.6b00597
  • ISSN: 0022-2623; 1520-4804
  • Keywords: Drug Discovery ; Molecular Medicine
  • Footnote: