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  1. Kany, Andreas M.; Sikandar, Asfandyar; Haupenthal, Jörg; Yahiaoui, Samir; Maurer, Christine K.; Proschak, Ewgenij; Köhnke, Jesko; Hartmann, Rolf W.

    Binding Mode Characterization and Early in Vivo Evaluation of Fragment-Like Thiols as Inhibitors of the Virulence Factor LasB from Pseudomonas aeruginosa

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    American Chemical Society (ACS), 2018

    Published in: ACS Infectious Diseases

  7. Yahiaoui, Samir; Voos, Katrin; Haupenthal, Jörg; Wichelhaus, Thomas A.; Frank, Denia; Weizel, Lilia; Rotter, Marco; Brunst, Steffen; Kramer, Jan S.; Proschak, Ewgenij; Ducho, Christian; Hirsch, Anna K. H.

    N-Aryl mercaptoacetamides as potential multi-target inhibitors of metallo-β-lactamases (MBLs) and the virulence factor LasB from Pseudomonas aeruginosa

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    Royal Society of Chemistry (RSC), 2021

    Published in: RSC Medicinal Chemistry

  8. Schönauer, Esther; Kany, Andreas M.; Haupenthal, Jörg; Hüsecken, Kristina; Hoppe, Isabel J.; Voos, Katrin; Yahiaoui, Samir; Elsässer, Brigitta; Ducho, Christian; Brandstetter, Hans; Hartmann, Rolf W.

    Discovery of a Potent Inhibitor Class with High Selectivity toward Clostridial Collagenases

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    American Chemical Society (ACS), 2017

    Published in: Journal of the American Chemical Society

  10. Jaouadi, Nadia Zaraî; Rekik, Hatem; Badis, Abdelmalek; Trabelsi, Sahar; Belhoul, Mouna; Yahiaoui, Amina Benkiar; Aicha, Houda Ben; Toumi, Abdessatar; Bejar, Samir; Jaouadi, Bassem

    Biochemical and Molecular Characterization of a Serine Keratinase from Brevibacillus brevis US575 with Promising Keratin-Biodegradation and Hide-Dehairing Activities

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    Public Library of Science (PLoS), 2013

    Published in: PLoS ONE

  11. Nordqvist, Anneli; Nilsson, Mikael T.; Lagerlund, Olof; Muthas, Daniel; Gising, Johan; Yahiaoui, Samir; Odell, Luke R.; Srinivasa, Bachally R.; Larhed, Mats; Mowbray, Sherry L.; Karlén, Anders

    Synthesis, biological evaluation and X-ray crystallographic studies of imidazo[1,2-a]pyridine-based Mycobacterium tuberculosis glutamine synthetase inhibitors

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    Royal Society of Chemistry (RSC), 2012

    Published in: MedChemComm

  12. Gising, Johan; Nilsson, Mikael T.; Odell, Luke R.; Yahiaoui, Samir; Lindh, Martin; Iyer, Harini; Sinha, Achyut M.; Srinivasa, Bachally R.; Larhed, Mats; Mowbray, Sherry L.; Karlén, Anders

    Trisubstituted Imidazoles as Mycobacterium tuberculosis Glutamine Synthetase Inhibitors

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    American Chemical Society (ACS), 2012

    Published in: Journal of Medicinal Chemistry

  13. Kaya, Cansu; Konstantinović, Jelena; Kany, Andreas M.; Andreas, Anastasia; Kramer, Jan S.; Brunst, Steffen; Weizel, Lilia; Rotter, Marco J.; Frank, Denia; Yahiaoui, Samir; Müller, Rolf; Hartmann, Rolf W.; Haupenthal, Jörg; Proschak, Ewgenij; Wichelhaus, Thomas A.; Hirsch, Anna K. H.

    N-Aryl Mercaptopropionamides as Broad-Spectrum Inhibitors of Metallo-β-Lactamases

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    American Chemical Society (ACS), 2022

    Published in: Journal of Medicinal Chemistry

  14. Konstantinović, Jelena; Yahiaoui, Samir; Alhayek, Alaa; Haupenthal, Jörg; Schönauer, Esther; Andreas, Anastasia; Kany, Andreas M.; Müller, Rolf; Koehnke, Jesko; Berger, Fabian K.; Bischoff, Markus; Hartmann, Rolf W.; Brandstetter, Hans; Hirsch, Anna K. H.

    N-Aryl-3-mercaptosuccinimides as Antivirulence Agents Targeting Pseudomonas aeruginosa Elastase and Clostridium Collagenases

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    American Chemical Society (ACS), 2020

    Published in: Journal of Medicinal Chemistry

  15. Jansson, Anna M.; Więckowska, Anna; Björkelid, Christofer; Yahiaoui, Samir; Sooriyaarachchi, Sanjeewani; Lindh, Martin; Bergfors, Terese; Dharavath, Shyamraj; Desroses, Matthieu; Suresh, Surisetti; Andaloussi, Mounir; Nikhil, Rautela; Sreevalli, Sharma; Srinivasa, Bachally R.; Larhed, Mats; Jones, T. Alwyn; Karlén, Anders; Mowbray, Sherry L.

    DXR Inhibition by Potent Mono- and Disubstituted Fosmidomycin Analogues

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    American Chemical Society (ACS), 2013

    Published in: Journal of Medicinal Chemistry

  16. Nilsson, Mikael T.; Krajewski, Wojciech W.; Yellagunda, Sujan; Prabhumurthy, Savitha; Chamarahally, Gayathri N.; Siddamadappa, Chandrasekharan; Srinivasa, Bachally R.; Yahiaoui, Samir; Larhed, Mats; Karlén, Anders; Jones, T. Alwyn; Mowbray, Sherry L.

    Structural Basis for the Inhibition of Mycobacterium tuberculosis Glutamine Synthetase by Novel ATP-Competitive Inhibitors

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    Elsevier BV, 2009

    Published in: Journal of Molecular Biology

  17. Schütz, Christian; Ho, Duy‐Khiet; Hamed, Mostafa Mohamed; Abdelsamie, Ahmed Saad; Röhrig, Teresa; Herr, Christian; Kany, Andreas Martin; Rox, Katharina; Schmelz, Stefan; Siebenbürger, Lorenz; Wirth, Marius; Börger, Carsten; Yahiaoui, Samir; Bals, Robert; Scrima, Andrea; Blankenfeldt, Wulf; Horstmann, Justus Constantin; Christmann, Rebekka; Murgia, Xabier; Koch, Marcus; Berwanger, Aylin; Loretz, Brigitta; Hirsch, Anna Katharina Herta; Hartmann, Rolf Wolfgang; [...]

    Pseudomonas aeruginosa Biofilm: A New PqsR Inverse Agonist Potentiates Tobramycin Efficacy to Eradicate Pseudomonas aeruginosa Biofilms (Adv. Sci. 12/2021)

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    Wiley, 2021

    Published in: Advanced Science

  18. Schütz, Christian; Ho, Duy‐Khiet; Hamed, Mostafa Mohamed; Abdelsamie, Ahmed Saad; Röhrig, Teresa; Herr, Christian; Kany, Andreas Martin; Rox, Katharina; Schmelz, Stefan; Siebenbürger, Lorenz; Wirth, Marius; Börger, Carsten; Yahiaoui, Samir; Bals, Robert; Scrima, Andrea; Blankenfeldt, Wulf; Horstmann, Justus Constantin; Christmann, Rebekka; Murgia, Xabier; Koch, Marcus; Berwanger, Aylin; Loretz, Brigitta; Hirsch, Anna Katharina Herta; Hartmann, Rolf Wolfgang; [...]

    A New PqsR Inverse Agonist Potentiates Tobramycin Efficacy to Eradicate Pseudomonas aeruginosa Biofilms

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    Wiley, 2021

    Published in: Advanced Science

  19. Rochais, Christophe; Lecoutey, Cédric; Gaven, Florence; Giannoni, Patrizia; Hamidouche, Katia; Hedou, Damien; Dubost, Emmanuelle; Genest, David; Yahiaoui, Samir; Freret, Thomas; Bouet, Valentine; Dauphin, François; Sopkova de Oliveira Santos, Jana; Ballandonne, Céline; Corvaisier, Sophie; Malzert-Fréon, Aurélie; Legay, Remi; Boulouard, Michel; Claeysen, Sylvie; Dallemagne, Patrick

    Novel Multitarget-Directed Ligands (MTDLs) with Acetylcholinesterase (AChE) Inhibitory and Serotonergic Subtype 4 Receptor (5-HT4R) Agonist Activities As Potential Agents against Alzheimer’s Disease: The Design of Donecopride

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    American Chemical Society (ACS), 2015

    Published in: Journal of Medicinal Chemistry

  20. Belaid, Brahim; Lamara Mahammed, Lydia; Drali, Ouardia; Oussaid, Aida Mohand; Touri, Nabila Souad; Melzi, Souhila; Dehimi, Abdelhak; Berkani, Lylia Meriem; Merah, Fatma; Larab, Zineb; Allam, Ines; Khemici, Ouarda; Kirane, Sonya Yasmine; Boutaba, Mounia; Belbouab, Reda; Bekkakcha, Hadjira; Guedouar, Assia; Chelali, Abdelhakim; Baamara, Brahim; Noui, Djamila; Baaziz, Hadda; Rezak, Radia; Azzouz, Sidi Mohamed; Aichaoui, Malika; [...]

    Inborn Errors of Immunity in Algerian Children and Adults: A Single-Center Experience Over a Period of 13 Years (2008–2021)

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    Frontiers Media SA, 2022

    Published in: Frontiers in Immunology