• Media type: E-Article
  • Title: Protein conformational flexibility modulates kinetics and thermodynamics of drug binding
  • Contributor: Amaral, Marta [Author]; Kokh, Daria B. [Author]; Wade, Rebecca C. [Author]
  • Published: 22 December 2017
  • Published in: Nature Communications ; 8(2017) Artikel-Nummer 2276, 14 Seiten
  • Language: English
  • DOI: 10.1038/s41467-017-02258-w
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  • Origination:
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  • Description: An understanding of the dynamics of drug binding and unbinding processes is important for drug discovery. Here, the authors give insights into the binding mechanism of small drug-like molecules to human Hsp90 by combining thermodynamics and kinetics studies as well as molecular dynamics simulations.
  • Access State: Open Access