• Media type: E-Article
  • Title: Fluorovinylsulfones and -Sulfonates as Potent Covalent Reversible Inhibitors of the Trypanosomal Cysteine Protease Rhodesain: Structure–Activity Relationship, Inhibition Mechanism, Metabolism, and In Vivo Studies
  • Contributor: Jung, Sascha; Fuchs, Natalie; Johe, Patrick; Wagner, Annika; Diehl, Erika; Yuliani, Tri; Zimmer, Collin; Barthels, Fabian; Zimmermann, Robert A.; Klein, Philipp; Waigel, Waldemar; Meyr, Jessica; Opatz, Till; Tenzer, Stefan; Distler, Ute; Räder, Hans-Joachim; Kersten, Christian; Engels, Bernd; Hellmich, Ute A.; Klein, Jochen; Schirmeister, Tanja
  • imprint: American Chemical Society (ACS), 2021
  • Published in: Journal of Medicinal Chemistry
  • Language: English
  • DOI: 10.1021/acs.jmedchem.1c01002
  • ISSN: 0022-2623; 1520-4804
  • Keywords: Drug Discovery ; Molecular Medicine
  • Origination:
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