• Media type: E-Article
  • Title: The Discovery of in Vivo Active Mitochondrial Branched-Chain Aminotransferase (BCATm) Inhibitors by Hybridizing Fragment and HTS Hits
  • Contributor: Bertrand, Sophie M.; Ancellin, Nicolas; Beaufils, Benjamin; Bingham, Ryan P.; Borthwick, Jennifer A.; Boullay, Anne-Bénédicte; Boursier, Eric; Carter, Paul S.; Chung, Chun-wa; Churcher, Ian; Dodic, Nerina; Fouchet, Marie-Hélène; Fournier, Charlène; Francis, Peter L.; Gummer, Laura A.; Herry, Kenny; Hobbs, Andrew; Hobbs, Clare I.; Homes, Paul; Jamieson, Craig; Nicodeme, Edwige; Pickett, Stephen D.; Reid, Iain H.; Simpson, Graham L.; [...]
  • imprint: American Chemical Society (ACS), 2015
  • Published in: Journal of Medicinal Chemistry
  • Language: English
  • DOI: 10.1021/acs.jmedchem.5b00313
  • ISSN: 0022-2623; 1520-4804
  • Keywords: Drug Discovery ; Molecular Medicine
  • Origination:
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