• Media type: E-Article
  • Title: Revisiting a challenging p53 binding site: a diversity-optimized HEFLib reveals diverse binding modes in T-p53C-Y220C
  • Contributor: Stahlecker, Jason; Klett, Theresa; Schwer, Martin; Jaag, Simon; Dammann, Marcel; Ernst, Larissa N.; Braun, Michael B.; Zimmermann, Markus O.; Kramer, Markus; Lämmerhofer, Michael; Stehle, Thilo; Coles, Murray; Boeckler, Frank M.
  • Published: Royal Society of Chemistry (RSC), 2022
  • Published in: RSC Medicinal Chemistry, 13 (2022) 12, Seite 1575-1586
  • Language: English
  • DOI: 10.1039/d2md00246a
  • ISSN: 2632-8682
  • Origination:
  • Footnote:
  • Description: Fragment screening of the challenging drug target T-p53-Y220C with our diversity optimized HEFLib leads to diverse reversible and covalent binding modes.
  • Access State: Open Access