• Medientyp: E-Artikel
  • Titel: Non-canonical activation of DAPK2 by AMPK constitutes a new pathway linking metabolic stress to autophagy
  • Beteiligte: Shiloh, Ruth; Gilad, Yuval; Ber, Yaara; Eisenstein, Miriam; Aweida, Dina; Bialik, Shani; Cohen, Shenhav; Kimchi, Adi
  • Erschienen: Springer Science and Business Media LLC, 2018
  • Erschienen in: Nature Communications, 9 (2018) 1
  • Sprache: Englisch
  • DOI: 10.1038/s41467-018-03907-4
  • ISSN: 2041-1723
  • Entstehung:
  • Anmerkungen:
  • Beschreibung: AbstractAutophagy is an intracellular degradation process essential for adaptation to metabolic stress. DAPK2 is a calmodulin-regulated protein kinase, which has been implicated in autophagy regulation, though the mechanism is unclear. Here, we show that the central metabolic sensor, AMPK, phosphorylates DAPK2 at a critical site in the protein structure, between the catalytic and the calmodulin-binding domains. This phosphorylation activates DAPK2 by functionally mimicking calmodulin binding and mitigating an inhibitory autophosphorylation, providing a novel, alternative mechanism for DAPK2 activation during metabolic stress. In addition, we show that DAPK2 phosphorylates the core autophagic machinery protein, Beclin-1, leading to dissociation of its inhibitor, Bcl-XL. Importantly, phosphorylation of DAPK2 by AMPK enhances DAPK2’s ability to phosphorylate Beclin-1, and depletion of DAPK2 reduces autophagy in response to AMPK activation. Our study reveals a unique calmodulin-independent mechanism for DAPK2 activation, critical to its function as a novel downstream effector of AMPK in autophagy.
  • Zugangsstatus: Freier Zugang