• Medientyp: E-Artikel
  • Titel: A New Cytotoxic Friedelane Acid – Pluricostatic Acid – and Other Compounds from the Leaves of Marila pluricostata
  • Beteiligte: Olmedo, Dionisio A.; López-Pérez, José L.; Del Olmo, Esther; Vásquez, Yelkaira; San Feliciano, Arturo; Gupta, Mahabir P.
  • Erschienen: MDPI AG, 2008
  • Erschienen in: Molecules, 13 (2008) 11, Seite 2915-2924
  • Sprache: Englisch
  • DOI: 10.3390/molecules13112915
  • ISSN: 1420-3049
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  • Beschreibung: Bioassay-guided fractionation of the dichloromethane extract of the leaves of Marila pluricostata led to the isolation of 2α,3β-dihydroxy-D:A-friedoolean-28-oic acid (pluricostatic acid), a new friedelane triterpenoid, (1), ten known triterpenoids and three sterols. Their chemical structures were elucidated through spectroscopic analysis. The less polar fractions, on GC/MS analysis and comparison with a MS library, resulted in the identification of twenty four sesquiterpenoids. The new triterpenoid acid 1 showed cytotoxicity against the MCF-7, H-460, and SF-268 human cancer cell lines with GI50 values from 1.2 to 3.3 μg/mL.
  • Zugangsstatus: Freier Zugang